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Home » Products » TIDEA screening compounds
TIDEA screening compounds
These molecules have TIDEA scores >9.5, and are more likely to exhibit submicromolar IC50s than lower-scoring molecules that bind to the same target. For more information on TIDEA, see www.focussynthesis.com/TIDEA
Catalog Number Structure FW Chemical Name and % Purity Please scroll down for more structures
Catalog #:   FS200062
CASRN:   170729-80-3
MFCD #:   MFCD08277635
534 APREPITANT
(Purity >97%)
In Stock: Price in US$
10
mg
100
mg
250
mg
1g 5g 20g 50g
195 995          
Catalog #:   FS005027
CASRN:   864685-46-1
MFCD #:   MFCD08062349
278 5-tert-Butyl-2-[2-(4-fluoro-phenoxy)-ethyl]2g,4-dihydro-pyrazol-3-one
(Purity >95%)
In Stock: Price in US$
10
mg
100
mg
250
mg
1g 5g 20g 50g
75 95 155        
Catalog #:   FS500002
CASRN:   
MFCD #:   MFCD18839169
470 (4-(Benzo[b]thiophen-3-ylsulfonyl)piperazin-1-yl)(3-(isothiazol-5-yl)phenyl)methanone
(Purity >%)
Special Order*: Price in US$
10
mg
100
mg
250
mg
1g 5g 20g 50g
  990          
Catalog #:   FS500035
CASRN:   
MFCD #:   MFCD18839181
418 3-(1-(Benzo[c][1,2,5]thiadiazol-4-ylsulfonyl)piperidin-4-yl)-6-fluorobenzo[d]isoxazole
(Purity >%)
Special Order*: Price in US$
10
mg
100
mg
250
mg
1g 5g 20g 50g
950 990          
Catalog #:   FS500025
CASRN:   
MFCD #:   MFCD18839178
444 (6-Bromoimidazo[1,2-a]pyrimidin-2-yl)(4-(6-fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)methanone
(Purity >%)
Special Order*: Price in US$
10
mg
100
mg
250
mg
1g 5g 20g 50g
  950 990        
Catalog #:   FS500052
CASRN:   
MFCD #:   MFCD18839193
403 (E)-tert-Butyl 2-(2-(4-methoxybenzyloxyimino)acetyl)-2,6-diazaspiro[3.4]octane-6-carboxylate
(Purity >%)
Special Order*: Price in US$
10
mg
100
mg
250
mg
1g 5g 20g 50g
890            
Catalog Number Structure FW Chemical Name and % Purity Please scroll down for more structures
Catalog #:   FS500072
CASRN:   
MFCD #:   MFCD18839191
334 tert-Butyl 2-(2-methoxyethylsulfonyl)-2,6-diazaspiro[3.4]octane-6-carboxylate
(Purity >%)
Special Order*: Price in US$
10
mg
100
mg
250
mg
1g 5g 20g 50g
980            
Catalog #:   FS500057
CASRN:   
MFCD #:   MFCD18839194
496 tert-Butyl 2-(3-(1,3-dioxoisoindolin-2-yloxy)propyl)-2,6-diazaspiro[3.4]octane-6-carboxylate hydrobromide
(Purity >%)
Special Order*: Price in US$
10
mg
100
mg
250
mg
1g 5g 20g 50g
980            
Catalog #:   FS500064
CASRN:   
MFCD #:   MFCD18839190
394 tert-Butyl 2-(4-acetylphenylsulfonyl)-2,6-diazaspiro[3.4]octane-6-carboxylate
(Purity >%)
Special Order*: Price in US$
10
mg
100
mg
250
mg
1g 5g 20g 50g
950            
Catalog #:   FS500068
CASRN:   
MFCD #:   MFCD18839192
466 tert-Butyl 2-(4-bromo-2-chlorophenylsulfonyl)-2,6-diazaspiro[3.4]octane-6-carboxylate
(Purity >%)
Special Order*: Price in US$
10
mg
100
mg
250
mg
1g 5g 20g 50g
890            
Catalog #:   FS500022
CASRN:   
MFCD #:   MFCD18839179
403 tert-Butyl 3-(4-(6-fluorobenzo[d]isoxazol-3-yl)piperidine-1-carbonyl)azetidine-1-carboxylate
(Purity >%)
Special Order*: Price in US$
10
mg
100
mg
250
mg
1g 5g 20g 50g
  950 990        
Catalog #:   FS500049
CASRN:   
MFCD #:   MFCD18839189
479 tert-Butyl 4-(3-(1-((1,3-dioxolan-2-yl)methyl)-1H-pyrazol-4-yl)phenylsulfonyl)piperazine-1-carboxylate
(Purity >%)
Special Order*: Price in US$
10
mg
100
mg
250
mg
1g 5g 20g 50g
890            
Catalog Number Structure FW Chemical Name and % Purity Please scroll down for more structures
Catalog #:   FS500017
CASRN:   
MFCD #:   MFCD18839172
447 tert-Butyl 4-(4-acetyl-N-(2,2-difluoroethyl)phenylsulfonamido)piperidine-1-carboxylate
(Purity >%)
Special Order*: Price in US$
10
mg
100
mg
250
mg
1g 5g 20g 50g
  990          
Catalog #:   FS500019
CASRN:   
MFCD #:   MFCD18839171
435 tert-Butyl 4-(N-(2,2-difluoroethyl)-4-methoxyphenylsulfonamido)piperidine-1-carboxylate
(Purity >%)
Special Order*: Price in US$
10
mg
100
mg
250
mg
1g 5g 20g 50g
  990          
Catalog #:   FS500012
CASRN:   
MFCD #:   MFCD18839173
397 tert-Butyl 4-(N-(2,2-difluoroethyl)-4H-furo[3,2-b]pyrrole-5-carboxamido)piperidine-1-carboxylate
(Purity >%)
Special Order*: Price in US$
10
mg
100
mg
250
mg
1g 5g 20g 50g
890 1490          
Catalog #:   FS500009
CASRN:   
MFCD #:   MFCD18839174
435 (2S,4S)-tert-Butyl 4-fluoro-2-(4-(6-fluorobenzo[d]isoxazol-3-yl)piperidine-1-carbonyl)pyrrolidine-1-carboxylate
(Purity >%)
Special Order*: Price in US$
10
mg
100
mg
250
mg
1g 5g 20g 50g
  990          
Catalog #:   FS500073
CASRN:   
MFCD #:   MFCD18839195
439 tert-Butyl 8-(2-(methoxycarbonyl)phenylsulfonyl)-2,8-diazaspiro[4.5]decane-2-carboxylate
(Purity >%)
Special Order*: Price in US$
10
mg
100
mg
250
mg
1g 5g 20g 50g
890            
Catalog #:   FS500011
CASRN:   
MFCD #:   MFCD18839175
530 (Z)-2,2-Difluoro-7-(4-(4-(6-fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)-4-oxobutoxyimino)-5H-[1,3]dioxolo[4,5-f]indol-6(7H)-one
(Purity >%)
Special Order*: Price in US$
10
mg
100
mg
250
mg
1g 5g 20g 50g
990            
Catalog Number Structure FW Chemical Name and % Purity Please scroll down for more structures
Catalog #:   FS500040
CASRN:   
MFCD #:   MFCD18839185
426 3-(1-(2-(Difluoromethoxy)phenylsulfonyl)piperidin-4-yl)-6-fluorobenzo[d]isoxazole
(Purity >%)
Special Order*: Price in US$
10
mg
100
mg
250
mg
1g 5g 20g 50g
  990          
Catalog #:   FS500043
CASRN:   
MFCD #:   MFCD10006850
302 2-(1-(3,4-Dimethylphenyl)-5-ethyl-1H-1,2,3-triazole-4-carboxamido)acetic acid
(Purity >%)
Special Order*: Price in US$
10
mg
100
mg
250
mg
1g 5g 20g 50g
495            
Catalog #:   FS500044
CASRN:   
MFCD #:   MFCD18839187
250 2-(1-((1,3-Dioxolan-2-yl)methyl)-1H-pyrazol-4-yl)-5-fluoropyrimidine
(Purity >%)
Special Order*: Price in US$
10
mg
100
mg
250
mg
1g 5g 20g 50g
  990          
Catalog #:   FS500047
CASRN:   
MFCD #:   MFCD18839188
349 1-((1,3-Dioxolan-2-yl)methyl)-4-(3-(azetidin-1-ylsulfonyl)phenyl)-1H-pyrazole
(Purity >%)
Special Order*: Price in US$
10
mg
100
mg
250
mg
1g 5g 20g 50g
  990          
Catalog #:   FS500021
CASRN:   
MFCD #:   MFCD18839177
342 6-Fluoro-3-(1-(2-methoxyethylsulfonyl)piperidin-4-yl)benzo[d]isoxazole
(Purity >%)
Special Order*: Price in US$
10
mg
100
mg
250
mg
1g 5g 20g 50g
  990          
Catalog #:   FS500041
CASRN:   
MFCD #:   MFCD18839186
411 6-Fluoro-3-(1-(isoquinolin-5-ylsulfonyl)piperidin-4-yl)benzo[d]isoxazole
(Purity >%)
Special Order*: Price in US$
10
mg
100
mg
250
mg
1g 5g 20g 50g
  990          
Catalog Number Structure FW Chemical Name and % Purity Please scroll down for more structures
Catalog #:   FS500031
CASRN:   
MFCD #:   
428 N-(3-(6-Fluorobenzo[d]isoxazol-3-yl)pentyl)-N-methylquinoline-8-sulfonamide
(Purity >%)
Special Order*: Price in US$
10
mg
100
mg
250
mg
1g 5g 20g 50g
  950 990        
Catalog #:   FS500001
CASRN:   
MFCD #:   MFCD18839168
383 (4-(3-(Isothiazol-5-yl)benzoyl)piperazin-1-yl)(thiophen-2-yl)methanone
(Purity >%)
At least 0.2 grams in stock
In Stock: Price in US$
10
mg
100
mg
250
mg
1g 5g 20g 50g
990            
Catalog #:   FS500005
CASRN:   
MFCD #:   MFCD18839170
498 (3-(Isothiazol-5-yl)phenyl)(4-(2-(trifluoromethoxy)phenylsulfonyl)piperazin-1-yl)methanone
(Purity >%)
Special Order*: Price in US$
10
mg
100
mg
250
mg
1g 5g 20g 50g
  990          
Catalog #:   FS500007
CASRN:   
MFCD #:   MFCD18839176
358 (4-(3-Methyl-[1,2,4]triazolo[4,3-a]pyridin-6-yl)phenyl)(piperazin-1-yl)methanone hydrochloride
(Purity >%)
Special Order*: Price in US$
10
mg
100
mg
250
mg
1g 5g 20g 50g
  990          
Catalog #:   FS200051
CASRN:   168273-06-1
MFCD #:   MFCD04034714
464 RIMONABANT
(Purity >97%)
Special Order*: Price in US$
10
mg
100
mg
250
mg
1g 5g 20g 50g
  495 995        


*Note concerning Special Order chemicals: these are made to order with a typical lead time of 6 weeks.
Minimum order sizes apply (usually 1 gram).
Prices are listed in the catalog for available quantities only.
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