These molecules have TIDEA scores >9.5, and are more likely to exhibit submicromolar IC50s than lower-scoring molecules that bind to the same target. For more information on TIDEA, see www.focussynthesis.com/TIDEA
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Structure |
FW |
Chemical Name and % Purity |
Click Price to Add to Shopping Cart |
|
Lead time: 2 weeks
|
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383 |
(4-(3-(Isothiazol-5-yl)benzoyl)piperazin-1-yl)(thiophen-2-yl)methanone (Purity >%)
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| Price in US dollars |
10 mg |
100 mg |
250 mg |
1g |
5g |
10g |
20g |
50g |
| |
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Lead time: IN STOCK
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278 |
5-tert-Butyl-2-[2-(4-fluoro-phenoxy)-ethyl]-2,4-dihydro-pyrazol-3-one (Purity >95%)
At least 0.58 grams in stock
|
| Price in US dollars |
10 mg |
100 mg |
250 mg |
1g |
5g |
10g |
20g |
50g |
| 75 |
95 |
155 |
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Lead time: Special Order*
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534 |
APREPITANT (Purity >97%)
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| Price in US dollars |
10 mg |
100 mg |
250 mg |
1g |
5g |
10g |
20g |
50g |
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Lead time: Special Order*
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418 |
3-(1-(Benzo[c][1,2,5]thiadiazol-4-ylsulfonyl)piperidin-4-yl)-6-fluorobenzo[d]isoxazole (Purity >%)
|
| Price in US dollars |
10 mg |
100 mg |
250 mg |
1g |
5g |
10g |
20g |
50g |
| 950 |
990 |
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Lead time: Special Order*
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 |
470 |
(4-(Benzo[b]thiophen-3-ylsulfonyl)piperazin-1-yl)(3-(isothiazol-5-yl)phenyl)methanone (Purity >%)
|
| Price in US dollars |
10 mg |
100 mg |
250 mg |
1g |
5g |
10g |
20g |
50g |
| |
990 |
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Lead time: Special Order*
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444 |
(6-Bromoimidazo[1,2-a]pyrimidin-2-yl)(4-(6-fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)methanone (Purity >%)
|
| Price in US dollars |
10 mg |
100 mg |
250 mg |
1g |
5g |
10g |
20g |
50g |
| |
950 |
990 |
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| |
Structure |
FW |
Chemical Name and % Purity |
Click Price to Add to Shopping Cart |
|
Lead time: Special Order*
|
 |
530 |
(Z)-2,2-Difluoro-7-(4-(4-(6-fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)-4-oxobutoxyimino)-5H-[1,3]dioxolo[4,5-f]indol-6(7H)-one (Purity >%)
|
| Price in US dollars |
10 mg |
100 mg |
250 mg |
1g |
5g |
10g |
20g |
50g |
| 990 |
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Lead time: Special Order*
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426 |
3-(1-(2-(Difluoromethoxy)phenylsulfonyl)piperidin-4-yl)-6-fluorobenzo[d]isoxazole (Purity >%)
|
| Price in US dollars |
10 mg |
100 mg |
250 mg |
1g |
5g |
10g |
20g |
50g |
| |
990 |
|
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Lead time: Special Order*
|
 |
302 |
2-(1-(3,4-Dimethylphenyl)-5-ethyl-1H-1,2,3-triazole-4-carboxamido)acetic acid (Purity >%)
|
| Price in US dollars |
10 mg |
100 mg |
250 mg |
1g |
5g |
10g |
20g |
50g |
| 495 |
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Lead time: Special Order*
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349 |
1-((1,3-Dioxolan-2-yl)methyl)-4-(3-(azetidin-1-ylsulfonyl)phenyl)-1H-pyrazole (Purity >%)
|
| Price in US dollars |
10 mg |
100 mg |
250 mg |
1g |
5g |
10g |
20g |
50g |
| |
990 |
|
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|
Lead time: 2 weeks
|
 |
250 |
2-(1-((1,3-Dioxolan-2-yl)methyl)-1H-pyrazol-4-yl)-5-fluoropyrimidine (Purity >%)
|
| Price in US dollars |
10 mg |
100 mg |
250 mg |
1g |
5g |
10g |
20g |
50g |
| |
990 |
|
|
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Lead time: Special Order*
|
 |
411 |
N-(3-(6-Fluorobenzo[d]isoxazol-3-yl)pentyl)-N-methylquinoline-8-sulfonamide (Purity >%)
|
| Price in US dollars |
10 mg |
100 mg |
250 mg |
1g |
5g |
10g |
20g |
50g |
| |
950 |
990 |
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|
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| |
Structure |
FW |
Chemical Name and % Purity |
Click Price to Add to Shopping Cart |
|
Lead time: Special Order*
|
 |
411 |
6-Fluoro-3-(1-(isoquinolin-5-ylsulfonyl)piperidin-4-yl)benzo[d]isoxazole (Purity >%)
|
| Price in US dollars |
10 mg |
100 mg |
250 mg |
1g |
5g |
10g |
20g |
50g |
| |
990 |
|
|
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Lead time: Special Order*
|
 |
342 |
6-Fluoro-3-(1-(2-methoxyethylsulfonyl)piperidin-4-yl)benzo[d]isoxazole (Purity >%)
|
| Price in US dollars |
10 mg |
100 mg |
250 mg |
1g |
5g |
10g |
20g |
50g |
| |
990 |
|
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|
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|
Lead time: Special Order*
|
 |
498 |
(3-(Isothiazol-5-yl)phenyl)(4-(2-(trifluoromethoxy)phenylsulfonyl)piperazin-1-yl)methanone (Purity >%)
|
| Price in US dollars |
10 mg |
100 mg |
250 mg |
1g |
5g |
10g |
20g |
50g |
| |
990 |
|
|
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Lead time: Special Order*
|
 |
358 |
(4-(3-Methyl-[1,2,4]triazolo[4,3-a]pyridin-6-yl)phenyl)(piperazin-1-yl)methanone hydrochloride (Purity >%)
|
| Price in US dollars |
10 mg |
100 mg |
250 mg |
1g |
5g |
10g |
20g |
50g |
| |
990 |
|
|
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Lead time: Special Order*
|
 |
464 |
RIMONABANT (Purity >97%)
|
| Price in US dollars |
10 mg |
100 mg |
250 mg |
1g |
5g |
10g |
20g |
50g |
| |
|
695 |
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Lead time: Special Order*
|
 |
447 |
tert-Butyl 4-(4-acetyl-N-(2,2-difluoroethyl)phenylsulfonamido)piperidine-1-carboxylate (Purity >%)
|
| Price in US dollars |
10 mg |
100 mg |
250 mg |
1g |
5g |
10g |
20g |
50g |
| |
990 |
|
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| |
Structure |
FW |
Chemical Name and % Purity |
Click Price to Add to Shopping Cart |
|
Lead time: Special Order*
|
 |
394 |
tert-Butyl 2-(4-acetylphenylsulfonyl)-2,6-diazaspiro[3.4]octane-6-carboxylate (Purity >%)
|
| Price in US dollars |
10 mg |
100 mg |
250 mg |
1g |
5g |
10g |
20g |
50g |
| 950 |
|
|
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Lead time: Special Order*
|
 |
466 |
tert-Butyl 2-(4-bromo-2-chlorophenylsulfonyl)-2,6-diazaspiro[3.4]octane-6-carboxylate (Purity >%)
|
| Price in US dollars |
10 mg |
100 mg |
250 mg |
1g |
5g |
10g |
20g |
50g |
| 890 |
|
|
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Lead time: Special Order*
|
 |
397 |
tert-Butyl 4-(N-(2,2-difluoroethyl)-4H-furo[3,2-b]pyrrole-5-carboxamido)piperidine-1-carboxylate (Purity >%)
|
| Price in US dollars |
10 mg |
100 mg |
250 mg |
1g |
5g |
10g |
20g |
50g |
| 890 |
1490 |
|
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Lead time: Special Order*
|
 |
435 |
tert-Butyl 4-(N-(2,2-difluoroethyl)-4-methoxyphenylsulfonamido)piperidine-1-carboxylate (Purity >%)
|
| Price in US dollars |
10 mg |
100 mg |
250 mg |
1g |
5g |
10g |
20g |
50g |
| |
990 |
|
|
|
|
|
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|
Lead time: Special Order*
|
 |
496 |
tert-Butyl 2-(3-(1,3-dioxoisoindolin-2-yloxy)propyl)-2,6-diazaspiro[3.4]octane-6-carboxylate hydrobromide (Purity >%)
|
| Price in US dollars |
10 mg |
100 mg |
250 mg |
1g |
5g |
10g |
20g |
50g |
| 980 |
|
|
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Lead time: Special Order*
|
 |
479 |
tert-Butyl 4-(3-(1-((1,3-dioxolan-2-yl)methyl)-1H-pyrazol-4-yl)phenylsulfonyl)piperazine-1-carboxylate (Purity >%)
|
| Price in US dollars |
10 mg |
100 mg |
250 mg |
1g |
5g |
10g |
20g |
50g |
| 890 |
|
|
|
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| |
Structure |
FW |
Chemical Name and % Purity |
Click Price to Add to Shopping Cart |
|
Lead time: Special Order*
|
 |
403 |
tert-Butyl 3-(4-(6-fluorobenzo[d]isoxazol-3-yl)piperidine-1-carbonyl)azetidine-1-carboxylate (Purity >%)
|
| Price in US dollars |
10 mg |
100 mg |
250 mg |
1g |
5g |
10g |
20g |
50g |
| |
950 |
990 |
|
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|
|
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Lead time: Special Order*
|
 |
435 |
(2S,4S)-tert-Butyl 4-fluoro-2-(4-(6-fluorobenzo[d]isoxazol-3-yl)piperidine-1-carbonyl)pyrrolidine-1-carboxylate (Purity >%)
|
| Price in US dollars |
10 mg |
100 mg |
250 mg |
1g |
5g |
10g |
20g |
50g |
| |
990 |
|
|
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Lead time: Special Order*
|
 |
403 |
(E)-tert-Butyl 2-(2-(4-methoxybenzyloxyimino)acetyl)-2,6-diazaspiro[3.4]octane-6-carboxylate (Purity >%)
|
| Price in US dollars |
10 mg |
100 mg |
250 mg |
1g |
5g |
10g |
20g |
50g |
| 890 |
|
|
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|
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Lead time: Special Order*
|
 |
439 |
tert-Butyl 8-(2-(methoxycarbonyl)phenylsulfonyl)-2,8-diazaspiro[4.5]decane-2-carboxylate (Purity >%)
|
| Price in US dollars |
10 mg |
100 mg |
250 mg |
1g |
5g |
10g |
20g |
50g |
| 890 |
|
|
|
|
|
|
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|
|
Lead time: Special Order*
|
 |
334 |
tert-Butyl 2-(2-methoxyethylsulfonyl)-2,6-diazaspiro[3.4]octane-6-carboxylate (Purity >%)
|
| Price in US dollars |
10 mg |
100 mg |
250 mg |
1g |
5g |
10g |
20g |
50g |
| 980 |
|
|
|
|
|
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